A-349,821

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A-349,821
A-349821.png
Systematic (IUPAC) name
(4'-[3-(2R,5R-dimethylpyrrolidin-1-yl)propoxy]biphenyl-4-yl)morpholin-4-ylmethanone
Identifiers
CAS Number 372513-99-0 N 556835-30-4 (trifluoroacetate salt)
PubChem CID: 9954017
IUPHAR/BPS 1217
ChemSpider 8129627 YesY
ChEMBL CHEMBL179702 YesY
Chemical data
Formula C26H34N2O3
Molecular mass 422.558
  • C[C@@H]1CC[C@H](N1CCCOC2=CC=C(C=C2)C3=CC=C(C=C3)C(=O)N4CCOCC4)C
  • InChI=1S/C26H34N2O3/c1-20-4-5-21(2)28(20)14-3-17-31-25-12-10-23(11-13-25)22-6-8-24(9-7-22)26(29)27-15-18-30-19-16-27/h6-13,20-21H,3-5,14-19H2,1-2H3/t20-,21-/m1/s1 YesY
  • Key:CFUHKRLMDNFZED-NHCUHLMSSA-N YesY
 NYesY (what is this?)  (verify)

A-349,821 is a potent and selective histamine H3 receptor antagonist[1] (or possibly an inverse agonist).[2] It has nootropic effects in animal studies,[3] although there do not appear to be any plans for clinical development at present and it is currently only used in laboratory research.

See also

H3 receptor antagonist

References

  1. ↑ Lua error in package.lua at line 80: module 'strict' not found.
  2. ↑ Lua error in package.lua at line 80: module 'strict' not found.
  3. ↑ Lua error in package.lua at line 80: module 'strict' not found.


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