DPI-3290

From Infogalactic: the planetary knowledge core
Jump to: navigation, search
DPI-3290
Structure of DPI-3290.png
Systematic (IUPAC) name
(+)-3-((αR)-α-((2S,5R)-4-Allyl-2,5-dimethyl-1-piperazinyl)-3-hydroxybenzyl)-N-(3-fluorophenyl)-N-methylbenzamide
Identifiers
CAS Number 182417-73-8 N
PubChem CID: 5242141
Chemical data
Formula C30H34FN3O2
Molecular mass 487.607 g/mol
  • OC1=CC=CC([C@@](C2=CC(C(N(C3=CC(F)=CC=C3)C)=O)=CC=C2)([H])N([C@@H](CN4CC=C)C)C[C@@H]4C)=C1
 NYesY (what is this?)  (verify)

DPI-3290 was discovered by Delta Pharmaceutical [1] and is a drug that is used in scientific research. It is a potent analgesic drug,[2] which produces little respiratory depression.[3]

DPI-3290 acts as an agonist at both μ- and δ-opioid receptor, with an IC50 of 6.2nM at μ and 1.0nM at δ.[4]

References

  1. ↑ US Patent 5552404 - Opioid compounds and methods for using same
  2. ↑ Lua error in package.lua at line 80: module 'strict' not found.
  3. ↑ Lua error in package.lua at line 80: module 'strict' not found.
  4. ↑ Lua error in package.lua at line 80: module 'strict' not found.


Retrieved from "https://infogalactic.com/w/index.php?title=DPI-3290&oldid=3435746"