Isamoltane

Isamoltane
Systematic (IUPAC) name
	1-(propan-2-ylamino)-3-(2-pyrrol-1-ylphenoxy)propan-2-ol
Identifiers
CAS Number	99740-06-4
ATC code	none
PubChem	CID: 127403
ChemSpider	113051
Chemical data
Formula	C16H22N2O2
Molecular mass	274.357 g/mol
	SMILES OC(CNC(C)C)COc1ccccc1n2cccc2 ;

Isamoltane (CGP-361A) is a drug used in scientific research. It acts as an antagonist at the β-adrenergic, 5-HT_1A, and 5-HT_1B receptors. It has about five times the potency for the 5-HT_1B receptor (21 nmol/l) over the 5-HT_1A receptor (112 nmol/l).^[1] It has anxiolytic effects in rodents.^[2]

References